In vitro anti-inflammatory activity of lignans isolated from Magnolia fargesii
  • Kim, Jae Yeon
  • Lim, Hyo Jin
  • Lee, Da Yeon
  • Kim, Ji Sun
  • Kim, Do Hee
  • ... Jeon, Raok
  • 외 3명
Citations

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84
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90

초록

The overproduction of nitric oxide (NO) and prostaglandin E-2 (PGE(2)) causes neurodegenerative diseases, such as Alzheimer's disease and Parkinson's disease. Four lignans, (+)-eudesmin (1), (+)-magnolin (2), (+)yangambin (3) and a new structure named as epimagnolin B (4) were isolated from Magnolia fargesii (Magnoliaceae) as the inhibitors of NO production in LPS-activated microglia. The most potent compound 4 inhibited the production of NO and PGE(2) and the expression of respective enzyme iNOS and COX-2 through the suppression of I-kappa B-alpha degradation and nuclear translocation of p65 subunit of NF-kappa B. (C) 2009 Published by Elsevier Ltd.

키워드

Magnolia fargesiiNitric oxideProstaglandin E-2MicrogliaNITRIC-OXIDE SYNTHASESFLOWER BUDSSELECTIVE INHIBITORFLOS-MAGNOLIAELIPOPOLYSACCHARIDESTEREOCHEMISTRYEXPRESSIONCYCLOOXYGENASE-2DERIVATIVESASSIGNMENT
제목
In vitro anti-inflammatory activity of lignans isolated from Magnolia fargesii
저자
Kim, Jae YeonLim, Hyo JinLee, Da YeonKim, Ji SunKim, Do HeeLee, Hwa JinKim, Hee DooJeon, RaokRyu, Jae-Ha
DOI
10.1016/j.bmcl.2008.11.103
발행일
2009-02-01
유형
Article
저널명
Bioorganic and Medicinal Chemistry Letters
19
3
페이지
937 ~ 940