유레아 및 티오유레아 유도체의 합성과 활성화된 대식세포의 NO 생성 저해효과

Synthesis of Urea and Thiourea Derivatives and Their Inhibitory Activities of NO Productionby Activated Macrophages
  • 김윤정; 
  • 천예진; 
  • 임효진; 
  • 류재하; 
  • 전라옥

초록

Several ureas and thioureas were designed and synthesized and their inhibitory activities of NO production in lipopolysaccharide-activated macrophages were evaluated. Among these compounds, indole-containing thiourea 6e was the most potent showing 17.4 μM of IC50 value.

키워드

urea; thiourea; nitric oxide; iNOS; indole; benzoxazole
제목
유레아 및 티오유레아 유도체의 합성과 활성화된 대식세포의 NO 생성 저해효과
제목 (타언어)
Synthesis of Urea and Thiourea Derivatives and Their Inhibitory Activities of NO Productionby Activated Macrophages
저자
김윤정; 천예진; 임효진; 류재하; 전라옥
발행일
2007-08
저널명
약 학 회 지
권
51
호
4
페이지
246 ~ 252