New estrogenic compounds isolated from Broussonetia kazinoki
  • Lee, Da Yeon
  • Kim, Do Hee
  • Lee, Hwa Jin
  • Lee, YoungJoo
  • Ryu, Kwang Hee
  • ... Song, Yun Seon
  • 외 2명
Citations

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26

초록

Two new and two known compounds were identified as estrogenic constituents from Broussonetia kazinoki. Their structures were elucidated as broussonin A (1), tupichinol C (2), kazinol U (3), and (+)-(2R) kazinol I (4). They showed estrogenic activity with ligand-binding activity of estrogen receptor, transcriptional activity of estrogen-responsive element-luciferase reporter genes. They also control the cellular gene expression levels of estrogen-responsive genes. Phytoestrogens from B. kazinoki may have beneficial effects in the treatment of menopausal symptoms. (C) 2010 Elsevier Ltd. All rights reserved.

키워드

Estrogen receptorPhytoestrogenBroussonetia kazinokiBREASTRECEPTORCANCERBETACONSTITUENTSMECHANISMSCOMPONENTFLAVANSALPHACELLS
제목
New estrogenic compounds isolated from Broussonetia kazinoki
저자
Lee, Da YeonKim, Do HeeLee, Hwa JinLee, YoungJooRyu, Kwang HeeJung, Bo-InSong, Yun SeonRyu, Jae-Ha
DOI
10.1016/j.bmcl.2010.04.064
발행일
2010-06-15
유형
Article
저널명
Bioorganic and Medicinal Chemistry Letters
20
12
페이지
3764 ~ 3767