Inhibition of lipopolysaccharide-induced inducible nitric oxide synthase and cyclooxygenase-2 expression by xanthanolides isolated from Xanthium strumarium
  • Yoon, Jeong Hoon
  • Lim, Hyo Jin
  • Lee, Hwa Jin
  • Kim, Hee-Doo
  • Jeon, Raok
  • 외 1명
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46
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50

초록

Three sesquiterpenoids, xanthatin (1), xanthinosin (2), and 4-oxo-bedfordia acid (3) were isolated from Xanthium strumarium as inhibitors of nitric oxide synthesis in activated microglia (IC50 values: 0.47, 11.2, 136.5 mu M, respectively). Compounds 1 and 2 suppressed the expression of iNOS and COX-2 and the activity of NF-kappa B through the inhibition of LPS-induced I-kappa B-alpha degradation in microglia. (C) 2008 Elsevier Ltd. All rights reserved.

키워드

nitric oxide synthasecyclooxygenaseXanthium strumariumsesquiterpenenuclear factor kappa BRAW 264.7 MACROPHAGESINFLAMMATORY RESPONSEINTERFERON-GAMMANERVOUS-SYSTEMBIOSYNTHESISDISEASESBRAINSTRATEGIESMICROGLIAINJURY
제목
Inhibition of lipopolysaccharide-induced inducible nitric oxide synthase and cyclooxygenase-2 expression by xanthanolides isolated from Xanthium strumarium
저자
Yoon, Jeong HoonLim, Hyo JinLee, Hwa JinKim, Hee-DooJeon, RaokRyu, Jae-Ha
DOI
10.1016/j.bmcl.2007.12.076
발행일
2008-03-15
유형
Article
저널명
Bioorganic and Medicinal Chemistry Letters
18
6
페이지
2179 ~ 2182